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Tiapamil hydrochloride
🥰Excellent
Catalog No. T13154Cas No. 57010-32-9
Alias Ro 11-1781 hydrochloride, ORE 5002 hydrochloride
Tiapamil hydrochloride (Ro 11-1781 hydrochloride) is a calcium channel blocker with antihypertensive activity and may be used in the study of angina and cardiovascular disease.
Tiapamil hydrochloride
🥰Excellent
Purity: 98.47%
Catalog No. T13154Alias Ro 11-1781 hydrochloride, ORE 5002 hydrochlorideCas No. 57010-32-9
Tiapamil hydrochloride (Ro 11-1781 hydrochloride) is a calcium channel blocker with antihypertensive activity and may be used in the study of angina and cardiovascular disease.
| Pack Size | Price | Availability | Quantity |
|---|---|---|---|
| 1 mg | $293 | In Stock | |
| 2 mg | $436 | In Stock | |
| 5 mg | $722 | In Stock | |
| 10 mg | $987 | In Stock | |
| 25 mg | $1,520 | In Stock | |
| 50 mg | $1,980 | In Stock |
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Purity:98.47%
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All TargetMol products are for research purposes only and cannot be used for human consumption. We do not provide products or services to individuals. Please comply with the intended use and do not use TargetMol products for any other purpose.Product Introduction
Bioactivity
Chemical Properties
| Description | Tiapamil hydrochloride (Ro 11-1781 hydrochloride) is a calcium channel blocker with antihypertensive activity and may be used in the study of angina and cardiovascular disease. |
| In vitro | Tiapamil hydrochloride is a novel calcium channel blocker with anti-anginal effects, which can be used to investigate the hemodynamics of patients with acute myocardial infarction[1]. |
| Alias | Ro 11-1781 hydrochloride, ORE 5002 hydrochloride |
| Molecular Weight | 592.16 |
| Formula | C26H38ClNO8S2 |
| Cas No. | 57010-32-9 |
| Smiles | Cl.O=S1(=O)CCCS(=O)(=O)C1(C2=CC=C(OC)C(OC)=C2)CCCN(C)CCC3=CC=C(OC)C(OC)=C3 |
| Relative Density. | no data available |
Storage & Solubility Information
| Storage | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice. |
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DMSO+30% PEG300+5% Tween 80+60% ddH2O. So your working solution concentration is 2 mg/mL。Mother liquor preparation method: 2 mg of drug dissolved in 50 μL DMSO (mother liquor concentration of 40 mg/mL), if you need to configure a concentration that exceeds the solubility of the product, please contact us first.
(mother liquor concentration of 40 mg/mL), if you need to configure a concentration that exceeds the solubility of the product, please contact us first.Preparation method for in vivo formula: Take 50 μL DMSO main solution, add 300 μLPEG300 mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLddH2O mix well and clarify
main solution, add 300 μLPEG300 mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLddH2O mix well and clarifyFor Reference Only. Please develop an appropriate dissolution method based on your laboratory animals and route of administration.
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